Using aminophylline for cellulite: home recipes and review of ready-made creams

What is cellulite

Cellulite is a pathology of adipose tissue caused by disturbances in the structure of cells. At first, “orange peel” is a barely noticeable cosmetic defect, expressed by tubercles and depressions on the skin. But if the problem is not solved in time, cellulite will actively develop and cause not only aesthetic, but also physical discomfort. The fact is that as the disease progresses, the affected areas become hard, lose sensitivity and turn blue. All this is fraught with tissue death, so under no circumstances should the “orange peel” appear.

To find out if you have cellulite, you need to squeeze the skin of your thigh.

Finding out if you have cellulite is simple: firmly squeeze the skin on your legs, buttocks or stomach with your fingers. If the surface of the epidermis is smooth, then there is no “orange peel”. Otherwise, you should resolve the problem as quickly as possible.

Ready-made anti-cellulite creams

Anti-orange peel products containing aminophylline are produced by several different companies. You should choose a specific one not only by price and brand, but also by skin type. For example, if the skin is dry, then creams are optimal for it, but for oily skin - gels. The most popular anti-cellulite products with aminophylline include:

• Evalar Turboslim . The cream is quite aggressive, causes a strong burning sensation when applied and therefore it can be diluted with a regular moisturizing or nourishing cream. Procedures with this product can hardly be called pleasant, but the result is impressive - after literally 5 applications, an increase in the elasticity of the skin and its smoothing are noted.
• Topical Aminophylline Gel . This remedy is most often used for applications that are placed specifically on problem areas of the body. The gel normalizes lipid metabolism, accelerating the breakdown of adipose tissue.
• Amilean . Available in gel form, it has maximum skin smoothing properties. According to testimonies from consumers and cosmetologists, this product can even get rid of stretch marks. There is only one significant drawback - the cost of the gel is very high and ranges from 3000 rubles (600 - 700 UAH) for a small tube.

What is Aminophylline?

Aminophylline is a drug originally intended to improve renal blood flow and treat bronchial asthma, bronchospasm and targeted vascular crises of atherosclerotic origin. The main active component of the product is the alkaloid theophylline. The latter is found in tea and coffee beans, but to make the drug it is synthesized artificially. In pharmacies the product can be found under the name “Eufilin”. The drug is sold in the form of ampoules and tablets.

Aminophylline is available in ampoules and tablets

How does Aminophylline fight cellulite?

In 1978, George Bay, a professor in the field of medicine, discovered a new property of Aminophylline - the ability to burn and break down subcutaneous fat. Thanks to this discovery, the drug began to be used in the fight against cellulite and excess weight. It should be borne in mind that the remedy is not a panacea and shows good results only with an integrated approach: proper nutrition, sufficient water intake, regular exercise, adequate sleep and keeping stressful situations to a minimum.

Aminophylline affects the skin as follows:

• Promotes the breakdown of fat deposits.
• It expels excess moisture from cells, thanks to which it successfully fights swelling.
• Relaxes muscles.
• Eliminates vascular spasms. As you know, one of the causes of cellulite is problems with the circulatory system.
• Improves metabolism at the cellular level.
• Accelerates blood circulation in tissues.
• Strongly heats the epidermis.
• Promotes gradual smoothing of textured, cellulite-affected skin.
• Prevents the formation of blood clots.
• Helps saturate epidermal cells with oxygen.

Aminophylline - what is it?

The principle of operation of the drug is explained by the action of the alkaloid theophylline, which relaxes the muscles, thereby smoothing the skin. The element belongs to the group of methylxanthines, which prevents the accumulation of adenosine monophosphate (cAMP). The enzyme reduces the activity of muscle proteins, thereby reducing muscle contraction and normalizing skin tone.

The alkaloid Theophylline is obtained synthetically, but it also occurs in nature. The alkaloid is found in coffee beans and tea leaves. Has all the effects of caffeine.

Simply put, aminophylline relaxes muscles, thereby reducing the likelihood of cramping. It also improves blood circulation and makes red blood cells more resistant to damage and deformation. Consequently, the drug relieves swelling and, due to the fact that blood circulates and nourishes the skin with oxygen, it looks better and the number of folds decreases.

Contraindications

We consider the drug Aminophylline as a means of combating cellulite, so we will only indicate side effects, indications and recommendations for use.

Aminophylline is not recommended for:

• severe hypertension;
• impaired functioning of the kidneys and liver;
• tachyarrhythmias;
• gastritis;
• epilepsy;
• disruption of the stomach and duodenum;
• presence of hemorrhagic stroke;
• retinal hemorrhage;
• aminophylline intolerance.

Side effects

When using the drug, side effects may occur in the form of:

• headaches;
• trembling of the whole body or its individual parts;
• increased arousal;
• tachycardia;
• sleep disorders;
• angina pectoris;
• arrhythmias;
• diarrhea;
• disturbances in the functioning of the stomach;
• itching;
• decreased appetite;
• rash;
• rapid breathing;
• sweating;
• hypoglycemia.

Aminophylline is contraindicated for pregnant women and those who are breastfeeding. The alkaloid theophylline can reach the fetus through the placenta. The concentration of the alkaloid is also observed in breast milk. Therefore, doctors recommend that all mothers who worry about their appearance take care of themselves after breastfeeding ends.

Contraindications

Aminophylline is a drug, so it has its own contraindications:

• arrhythmia,
• respiratory tract diseases,
• acute and chronic form of renal failure,
• varicose veins,
• stomach ulcer,
• hormonal disbalance,
• prostate adenoma,
• high blood pressure,
• individual intolerance,
• high pressure,
• alcoholism,
• disruption of the normal functioning of the thyroid gland.

Useful properties of Eufillin against cellulite

In the photo, Eufillin for cellulite. Price - from 12 rubles. for 30 tablets.

Eufillin is a medicine that belongs to the category of bronchodilators. The active ingredient is aminophylline. In simple terms, it affects blood vessels, dilating them. Thanks to this, problems in the functioning of the respiratory system are solved. The drug is also used to treat vascular spasms.

Eufillin has several main effects:

• vasodilation;
• muscle relaxation;
• improved blood flow.

The effect on cellulite is that the skin begins to heat up. Eufillin is used externally. Under its influence, blood flow accelerates, while a person feels a pleasant tingling and warmth. This means that work begins inside the fatty tissues.

Along with the activation of processes, fat cells are broken down, and the removal of toxins and excess fluid begins. This leads to a reduction in swelling and a skin tightening effect.

Eufillin is available in tablets of 150 mg of active ingredient. Ampoules are also sold - 5 and 10 ml. They contain a solution of 2.4% and 24%. In the first case, the drug is intended for intravenous administration, in the second - intramuscular.

Eufillin against cellulite is an inexpensive medicine. Prices for the drug are within the following limits:

• 30 tablets - from 12 rubles;
• solution, 2.4%, 10 ampoules of 10 ml - from 66 rubles.

Side effects after use

The following side effects may occur when using Aminophylline:

• noise in ears,
• increased fatigue,
• high blood pressure,
• headache,
• darkening in the eyes,
• itching,
• redness,
• rash,
• burning.

If your skin turns red, don't be alarmed. This may be a sign of blood flow to the treated area. However, if the redness does not go away for a long time, you should consult a doctor.

Making cream at home

You can test the anti-cellulite effect of the substance by preparing the cream yourself. For this you will need pure aminophylline or its analogue aminophylline. Ampoules are sold in pharmacies and are much cheaper than ready-made products. Dimexide is often added to recipes because it accelerates the transport of aminophylline into tissues. To prepare homemade creams, it is important to follow the correct dosage of ingredients:

• cellulite cream can be enriched with aminophylline by adding 1 ampoule to 50 g of cosmetic product;
• mix the following ingredients in a 1:1 ratio: aminophylline (10 ml), vegetable oil, Vaseline, baby cream and apply to the skin. The resulting mixture is well absorbed and does not cause irritation to the skin;
• dissolve 2 mg of dimexide in 1 ampoule of aminophylline, apply to problem areas;
• combine 1 ampoule of aminophylline, dimexide (10 ml) with regular body cream (40 g).

Precautionary measures

To avoid side effects when using Aminophylline, you should adhere to the following precautions:

• Do not rub more than one tablet or 5 ml of the drug into the skin at a time (per 70 kg of body weight).
• Be sure to do an allergy test before using the product: apply a little Aminophylline to your wrist or elbow. If after a day there is no irritation, feel free to use the drug.
• Do not use expired product as this may cause unexpected consequences.
• Do not apply the drug or formulations based on it to irritated or damaged skin.
• If you notice signs of individual intolerance to the product (irritation, rash, etc.), stop using the product immediately.
• Drink as much fluid as possible during any procedure using Aminophylline. In this way you protect the urinary system from retention of the drug in it.

Eufillin, 30 pcs., 150 mg, tablets

Pharmaceutical group: bronchodilator. Pharmaceutical action: Eufillin is a bronchodilator, a xanthine derivative; inhibits phosphodiesterase, increases the accumulation of cyclic adenosine monophosphate in tissues, blocks adenosine (purine) receptors; reduces the flow of calcium ions through the channels of cell membranes, reduces the contractile activity of smooth muscles. Relaxes the bronchial muscles, increases mucociliary clearance, stimulates contraction of the diaphragm, improves the function of the respiratory and intercostal muscles, stimulates the respiratory center, increases its sensitivity to carbon dioxide and improves alveolar ventilation, which ultimately leads to a decrease in the severity and frequency of apnea episodes. By normalizing respiratory function, it helps saturate the blood with oxygen and reduce the concentration of carbon dioxide. It has a stimulating effect on the activity of the heart, increases the strength and number of heart contractions, increases coronary blood flow and myocardial oxygen demand. Reduces the tone of blood vessels (mainly those of the brain, skin and kidneys). It has a peripheral venodilating effect, reduces pulmonary vascular resistance, and reduces pressure in the “lesser” circulation. Increases renal blood flow and has a moderate diuretic effect. Expands extrahepatic bile ducts. Inhibits platelet aggregation (suppresses platelet activating factor and PgE2 alpha), increases the resistance of red blood cells to deformation (improves the rheological properties of blood), reduces thrombus formation and normalizes microcirculation. It has a tocolytic effect, increases the acidity of gastric juice. When used in large doses, it has an enileptogenic effect. Pharmacokinetics: After oral administration, it is quickly and completely absorbed, bioavailability is 90-100%. Food reduces the rate of absorption without affecting its magnitude (large volumes of liquid and proteins speed up the process). The higher the dose taken, the lower the absorption rate. The time to reach Cmax is 1-2 hours. Vd is in the range of 0.3-0.7 l/kg (30-70% of the “ideal” body weight), on average 0.45 l/kg. The connection with plasma proteins in adults is 60%, in patients with liver cirrhosis - 36%. Penetrates into breast milk (10% of the dose taken), through the placental barrier (the concentration in the fetal blood serum is slightly higher than in the maternal serum). Aminophylline exhibits bronchodilating properties in concentrations of 10-20 mcg/ml. Concentrations above 20 mg/ml are toxic. The stimulating effect on the respiratory center is realized at a lower content of the drug in the blood of 5-10 mcg/ml. Metabolized at physiological pH values ​​with the release of free theophylline, which is further metabolized in the liver with the participation of several cytochrome P450 isoenzymes. As a result, 1, 3-dimethyluric acid (45-55%) is formed, which has pharmacological activity, but is 1-5 times inferior to theophylline. Caffeine is an active metabolite and is formed in small quantities. In children over 3 years of age and in adults (unlike younger children), the phenomenon of caffeine accumulation is absent. T1/2 in children over 6 months – 3.7 hours; in adults – 8.7 hours; for “smokers” (20-40 cigarettes per day) - 4-5 hours (after quitting smoking, pharmacokinetics normalize after 3-4 months); in adults with chronic obstructive pulmonary disease, pulmonary heart disease and pulmonary heart failure - over 24 hours. Excreted by the kidneys.

How aminophylline fights “orange peel”

Anti-cellulite cream with aminophylline will help you quickly get rid of the hated bumps on the skin. The drug gained popularity recently, and has become known since the end of the twentieth century. Initially it was used to treat pulmonary and bronchial diseases. It was not immediately known that the medicine could affect the subcutaneous fat layer.

The action of amyophylline is as follows:

• Penetrates deep into the fat layer;
• Saturates tissues with oxygen;
• Provokes the breakdown of fat cells;
• Improves blood flow, lymphatic drainage, helps eliminate tissue swelling, irritates the skin.

Be sure to read: BCAA amino acid complex from the manufacturer Dymatize Nutrition

Euphylline (another name for the drug) contains theophylline, an artificial alkaloid. It can penetrate the skin either through injections or through the outer layer of the epidermis. The substance is able to relax the muscles of the muscles, due to which the skin becomes smooth and elastic.

Store and pharmacy cosmetics

Modern manufacturers offer a large selection of gels and creams with Aminophylline against cellulite. Let's look at the most popular and effective ones.

Advice! When choosing anti-cellulite cosmetics, be guided by your skin type. Creams are suitable for dry skin, and light gels for oily skin.